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Ngwaahịa

Cytisine

Nkọwa dị mkpirikpi:

Gịnị bụ isi iyi nke Cytisine?

● A na-esikarị n’osisi ahịhịa amịpụta ahịhịa, dị ka ahịhịa, agwa ilu, na cassia ọhịa. Mkpụrụ ma ọ bụ osisi niile nke osisi ndị a bara ụba na plantain.

●N'oge usoro mmịpụta, a na-ekewa metronidine ma mee ka ọ dị ọcha dị ka ihe ezubere iche, na akụkụ bụ isi nke ngwaahịa ikpeazụ bụ metronidine.


Nkọwa ngwaahịa

Mkpado ngwaahịa

Ihe omuma nke Cytisine

Ozi ndị bụ isi:
Usoro ọgwụ: C₁₁H₁₄N₂O
Arọ molikula: 190.24
Ọdịdị: Grayish-acha ọcha ruo odo-aja aja crystalline siri ike, ma ọ bụ orthorhombic prismatic ntụ ntụ
Ebe mgbaze: 154-156 ℃
Nsi: O nwere ụfọdụ nsi na ekwesịrị iji nlezianya mee ya

Gịnị bụ pharmacological mmetụta nke Cytsin?

● Mmasị iku ume: Mmetụta ọ na-enwe n'usoro iku ume yiri nke nicotine. Ọ nwere ike na-akpali akpali nke iku ume center, welie omimi na ugboro nke iku ume, na mmetụta ya nke na-akpali iku ume dị ike karịa nke otu dose nke phellodenine.

● Mgbochi obi mgbawa: Ọ nwere ike ibelata mgbakasị ahụ na ịrụ ọrụ nke myocardial, ngwa ngwa obi, na-egbochi myocardial contractility, na ịgbatị oge mgbakasị ahụ. Enwere ike iji ya na-agwọ tachycardia ventricular na palpitations na-arụ ọrụ

● Ọrụ ndị ọzọ: Nnyocha e mere n'oge na-adịbeghị anya egosiwo na ọ nwekwara ọtụtụ ihe omume ọgwụ dị ka ọrịa nje na-alụso ọrịa ọgụ, mgbochi ọnya, ịba ụba mkpụrụ ndụ ọbara ọcha, na mgbochi ọrịa cancer. N'ihe banyere ọrụ mgbochi ọrịa cancer, ọ nwere ike ịkpata apoptosis nke mkpụrụ ndụ kansa ma ejiri ya mee ihe n'ọtụtụ ebe iji gbochie mgbasa nke mkpụrụ ndụ tumor dị iche iche.

Gịnị bụ kpọmkwem mmetụta anwansi nke Cytsin?

● Mmetụta ịkwụsị ịṅụ sịga: Plantarine bụ alkaloid nke nwere njikọ dị elu na nicotine-acetylcholine receptor. Ọ nwere ike rụọ ọrụ dị ka onye agonist mpaghara na-ahọrọ, na-ebelata ịdabere na nicotine ndị na-ese siga, na-ebelata agụụ ise siga, na ibelata ogo mgbaàmà nkwụsị nicotine.

● Mmetụta ume iku ume: Mmetụta metronidine na usoro iku ume yiri nke nicotine. Ọ nwere ike na-akpali akpali nke iku ume etiti, na-eme ka omimi na ugboro nke iku ume

● Mmetụta mgbochi arrhythmic: Clindamine nwere ike ibelata mgbakasị myocardial na conductivity, obi na-adịghị ngwa ngwa, na-egbochi myocardial contractility, na-agbatị oge nkwụsịtụ, si otú a na-eji agwọ tachycardia ventricular na palpitations na-arụ ọrụ.

● Mmetụta na-egbochi ọrịa cancer: Plantarine nwere ike ịkpata apoptosis nke mkpụrụ ndụ kansa ma gbochie mmụba nke mkpụrụ ndụ tumor dị iche iche n'ihe gbasara ọrụ mgbochi ọrịa cancer.

● Ọrụ ndị ọzọ: Clindamine na-enwekwa mmetụta nke nje na-alụso ọrịa ọgụ, na-egbochi ọnya ọnya, ịba ụba nke mkpụrụ ndụ ọbara ọcha, na-eme ka ọrụ ọgụgụ isi dịkwuo mma, na-egbochi ịda mbà n'obi.

Kpọtụrụ: Judy Guo
WhatsApp/anyị kparịta ụka:+86-18292852819
E-mail:sales3@xarainbow.com


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